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                原料药及中间体服务

                吉林ξ 天衡原料药和中间体生产基地位于河南省邓州市工业园区南阳天衡制药厂,车间占地1万平米,各类型反应釜40余台。依托北京天衡药物研究院有限公司产品的研发 ,已完成》小试品种有100多个,目前工业化规模生产13个品种,产品质量达到国际高水平。产品出口日本ξ、印度、东南亚和欧洲部分国家。


                原料药及中间体服务产品目录



                产品名称Product nameCAS登记号(CAS No.)标准Specification结构式Structural Formula
                伏格列波糖及中间体
                Voglibose & Intermediates
                伏格列波糖
                Voglibose
                83480-29-9JP16
                IP
                In house
                 01
                2,3,4,6-四-O-苄基-α-D-葡萄糖
                2,3,4,6-Tetra-O-benzyl-α-D-glucopyranose
                4132-28-9
                6564-72-3
                ≥99%
                In house
                 02
                (2R,3S,4S,5S)-5-羟基-2,3,4-三 (苄氧基)-5-[(苄氧基)甲基]-环己酮 (2R,3S,4S,5S)-5-Hydroxy-2,3,4-tris (phenylmethoxy)-5-[(phenylmethoxy)methyl]-cyclohexanone115250-38-9≥99%
                In house
                 03
                四苄基伏格列波糖
                Tetra-Benzyl-Voglibose
                115250-39-0≥99%
                In house
                 04
                盐酸吉西他滨中间体Gemcitabine Hydrochloride Intermediate2-脱氧-2,2二氟-戊呋喃糖-1-酮- 3,5-二苯甲酸酯(T6) 2-Deoxy-2,2-difluoro-D-erythro-pentafuranous-1-ulose-3,5-dibenzoate122111-01-7≥99%
                In house
                 05
                帕利哌酮及中间体
                Paliperidone & Intermediates
                帕利哌酮
                Paliperidone
                144598-75-4≥99%
                In house
                 06
                帕利哌酮棕榈酸酯
                Paliperidone Palmitate
                199739-10-1≥99%
                In house
                 07
                3-(2-氯乙基)-6,7,8,9-四氢-9-羟基-2-甲基-4H-吡啶并[1,2-a]嘧啶-4-酮3-(2-Chloroethyl)-6,7,8,9-tetrahydro-9-hydroxy-2-methyl-4H-pyrido[1,2-a]pyrimidin-4-one130049-82-0≥99%
                In house
                 08
                6-氟-3-哌啶-4-基-1,2-苯并异噁唑盐酸盐
                6-Fluoro-3-(4-piperidinyl)-1,2-
                benzisoxazole hydrochloride
                84163-13-3≥99%
                In house
                 09
                盐酸厄洛替尼中间体
                Erlotinib Hydrochloride
                Intermediates
                6,7-双(甲氧基乙氧①基)喹唑啉酮
                6,7-Bis-(2-methoxyethoxy)-4(3H)-quinazolinone
                179688-29-0≥99%
                In house
                 10
                阿加曲班及中间体Argatroban &
                Intermediate
                阿加曲班
                Argatroban Hydrate
                74863-84-6≥99%
                In house
                 11
                (2R,4R)-4-甲基-2-哌啶甲酸乙酯
                Ethyl (2R,4R)-4-methyl-2-piperidinecarboxylate
                74892-82-3≥99%
                     In house
                 12
                帕布昔利布及中间体Palbociclib & Intermediates帕布昔利布(帕博西尼)
                Palbociclib
                571190-30-2≥99%
                In house
                 13
                4-(6-氨基吡啶-3-基)哌嗪-1-羧酸叔丁酯
                4-(6-Aminopyridin-3-yl)piperazine-1-carboxylic acid tert-butyl este
                571188-59-5≥99%
                In house
                 14
                6-溴-2-氯-8-环戊基-5-甲基-吡啶并[2,3-D]嘧啶-7(8H)-酮6-bromo-2-chloro-8-cyclopentyl-5-Methylpyrido[2,3-d]pyriMidin-7(8H)-one1016636-76-2≥99%
                In house
                 15
                奥格列汀Omarigliptin & IntermediatesN-[(2R,3S)-2-(2,5-二氟苯基)四氢-5-氧代-2H-吡喃-3-基]氨基甲酸叔丁酯N-[(2R,3S)-2-(2,5-Difluorophenyl)tetrahydro-5-oxo-2H-pyran-3-yl]carbamic acid 1,1-dimethylethyl ester951127-25-6≥99%
                In house
                 16
                2-(甲基磺酰基)-2,4,5,6-四氢吡咯并[3,4-c]吡唑苯⊙磺酸盐
                2,4,5,6-Tetrahydro-2-(methylsulfonyl)pyrrolo[3,4-c]pyrazole benzenesulfonate
                1280210-80-1≥99%
                In house
                 17