原料药及中间体服务
吉林ξ 天衡原料药和中间体生产基地位于河南省邓州市工业园区南阳天衡制药厂,车间占地1万平米,各类型反应釜40余台。依托北京天衡药物研究院有限公司产品的研发 ,已完成》小试品种有100多个,目前工业化规模生产13个品种,产品质量达到国际高水平。产品出口日本ξ、印度、东南亚和欧洲部分国家。
原料药及中间体服务产品目录
产品名称Product name | CAS登记号(CAS No.) | 标准Specification | 结构式Structural Formula | |
伏格列波糖及中间体 Voglibose & Intermediates | 伏格列波糖 Voglibose | 83480-29-9 | JP16 IP In house | ![]() |
2,3,4,6-四-O-苄基-α-D-葡萄糖 2,3,4,6-Tetra-O-benzyl-α-D-glucopyranose | 4132-28-9 6564-72-3 | ≥99% In house | ![]() | |
(2R,3S,4S,5S)-5-羟基-2,3,4-三 (苄氧基)-5-[(苄氧基)甲基]-环己酮 (2R,3S,4S,5S)-5-Hydroxy-2,3,4-tris (phenylmethoxy)-5-[(phenylmethoxy)methyl]-cyclohexanone | 115250-38-9 | ≥99% In house | ![]() | |
四苄基伏格列波糖 Tetra-Benzyl-Voglibose | 115250-39-0 | ≥99% In house | ![]() | |
盐酸吉西他滨中间体Gemcitabine Hydrochloride Intermediate | 2-脱氧-2,2二氟-戊呋喃糖-1-酮- 3,5-二苯甲酸酯(T6) 2-Deoxy-2,2-difluoro-D-erythro-pentafuranous-1-ulose-3,5-dibenzoate | 122111-01-7 | ≥99% In house | ![]() |
帕利哌酮及中间体 Paliperidone & Intermediates | 帕利哌酮 Paliperidone | 144598-75-4 | ≥99% In house | ![]() |
帕利哌酮棕榈酸酯 Paliperidone Palmitate | 199739-10-1 | ≥99% In house | ![]() | |
3-(2-氯乙基)-6,7,8,9-四氢-9-羟基-2-甲基-4H-吡啶并[1,2-a]嘧啶-4-酮3-(2-Chloroethyl)-6,7,8,9-tetrahydro-9-hydroxy-2-methyl-4H-pyrido[1,2-a]pyrimidin-4-one | 130049-82-0 | ≥99% In house | ![]() | |
6-氟-3-哌啶-4-基-1,2-苯并异噁唑盐酸盐 6-Fluoro-3-(4-piperidinyl)-1,2- benzisoxazole hydrochloride | 84163-13-3 | ≥99% In house | ![]() | |
盐酸厄洛替尼中间体 Erlotinib Hydrochloride Intermediates | 6,7-双(甲氧基乙氧①基)喹唑啉酮 6,7-Bis-(2-methoxyethoxy)-4(3H)-quinazolinone | 179688-29-0 | ≥99% In house | ![]() |
阿加曲班及中间体Argatroban & Intermediate | 阿加曲班 Argatroban Hydrate | 74863-84-6 | ≥99% In house | ![]() |
(2R,4R)-4-甲基-2-哌啶甲酸乙酯 Ethyl (2R,4R)-4-methyl-2-piperidinecarboxylate | 74892-82-3 | ≥99% In house | ![]() | |
帕布昔利布及中间体Palbociclib & Intermediates | 帕布昔利布(帕博西尼) Palbociclib | 571190-30-2 | ≥99% In house | ![]() |
4-(6-氨基吡啶-3-基)哌嗪-1-羧酸叔丁酯 4-(6-Aminopyridin-3-yl)piperazine-1-carboxylic acid tert-butyl este | 571188-59-5 | ≥99% In house | ![]() | |
6-溴-2-氯-8-环戊基-5-甲基-吡啶并[2,3-D]嘧啶-7(8H)-酮6-bromo-2-chloro-8-cyclopentyl-5-Methylpyrido[2,3-d]pyriMidin-7(8H)-one | 1016636-76-2 | ≥99% In house | ![]() | |
奥格列汀Omarigliptin & Intermediates | N-[(2R,3S)-2-(2,5-二氟苯基)四氢-5-氧代-2H-吡喃-3-基]氨基甲酸叔丁酯N-[(2R,3S)-2-(2,5-Difluorophenyl)tetrahydro-5-oxo-2H-pyran-3-yl]carbamic acid 1,1-dimethylethyl ester | 951127-25-6 | ≥99% In house | ![]() |
2-(甲基磺酰基)-2,4,5,6-四氢吡咯并[3,4-c]吡唑苯⊙磺酸盐 2,4,5,6-Tetrahydro-2-(methylsulfonyl)pyrrolo[3,4-c]pyrazole benzenesulfonate | 1280210-80-1 | ≥99% In house | ![]() |